DE69518323T2 - Oxaborole und deren salze, und deren verwendung als biozide - Google Patents

Oxaborole und deren salze, und deren verwendung als biozide

Info

Publication number
DE69518323T2
DE69518323T2 DE69518323T DE69518323T DE69518323T2 DE 69518323 T2 DE69518323 T2 DE 69518323T2 DE 69518323 T DE69518323 T DE 69518323T DE 69518323 T DE69518323 T DE 69518323T DE 69518323 T2 DE69518323 T2 DE 69518323T2
Authority
DE
Germany
Prior art keywords
pct
oxaborole
biocides
salts
date dec
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69518323T
Other languages
English (en)
Other versions
DE69518323D1 (de
Inventor
William Austin
Juan Kneale
Jelf Crowley
Martin CLOUGH
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Avecia Ltd
Original Assignee
Avecia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Avecia Ltd filed Critical Avecia Ltd
Application granted granted Critical
Publication of DE69518323D1 publication Critical patent/DE69518323D1/de
Publication of DE69518323T2 publication Critical patent/DE69518323T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/0008—Organic ingredients according to more than one of the "one dot" groups of C08K5/01 - C08K5/59
    • C08K5/0058—Biocides
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09D—COATING COMPOSITIONS, e.g. PAINTS, VARNISHES OR LACQUERS; FILLING PASTES; CHEMICAL PAINT OR INK REMOVERS; INKS; CORRECTING FLUIDS; WOODSTAINS; PASTES OR SOLIDS FOR COLOURING OR PRINTING; USE OF MATERIALS THEREFOR
    • C09D5/00—Coating compositions, e.g. paints, varnishes or lacquers, characterised by their physical nature or the effects produced; Filling pastes
    • C09D5/14—Paints containing biocides, e.g. fungicides, insecticides or pesticides
DE69518323T 1994-06-09 1995-05-26 Oxaborole und deren salze, und deren verwendung als biozide Expired - Fee Related DE69518323T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9411587A GB9411587D0 (en) 1994-06-09 1994-06-09 Compound, composition and use
PCT/GB1995/001206 WO1995033754A1 (en) 1994-06-09 1995-05-26 Oxaboroles and salts thereof, and their use as biocides

Publications (2)

Publication Number Publication Date
DE69518323D1 DE69518323D1 (de) 2000-09-14
DE69518323T2 true DE69518323T2 (de) 2001-02-01

Family

ID=10756481

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69518323T Expired - Fee Related DE69518323T2 (de) 1994-06-09 1995-05-26 Oxaborole und deren salze, und deren verwendung als biozide

Country Status (14)

Country Link
US (1) US5880188A (de)
EP (1) EP0765331B1 (de)
JP (1) JPH10500983A (de)
KR (1) KR970703349A (de)
CN (1) CN1068005C (de)
AT (1) ATE195316T1 (de)
AU (1) AU681291B2 (de)
BR (1) BR9507966A (de)
CA (1) CA2190155A1 (de)
DE (1) DE69518323T2 (de)
GB (1) GB9411587D0 (de)
NO (1) NO965235L (de)
TW (1) TW368397B (de)
WO (1) WO1995033754A1 (de)

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US6184363B1 (en) 1997-06-13 2001-02-06 Northwestern University Inhibitors of β-lactamases and uses therefor
US7465836B2 (en) * 2003-06-16 2008-12-16 Anacor Pharmaceuticals, Inc. Hydrolytically-resistant boron-containing therapeutics and methods of use
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NZ598441A (en) * 2005-02-16 2013-07-26 Anacor Pharmaceuticals Inc Boron-containing small molecules
WO2007078340A2 (en) 2005-12-30 2007-07-12 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
CN102532180B (zh) * 2005-12-30 2016-06-29 安纳考尔医药公司 含硼的小分子
DK2719388T3 (da) * 2006-02-16 2019-05-13 Anacor Pharmaceuticals Inc Borholdige små molekyler som antiinflammatoriske midler
US20070197388A1 (en) * 2006-02-22 2007-08-23 Buckman Laboratories International, Inc. Haloperoxidase treatment to control algae
RU2486914C2 (ru) * 2006-03-16 2013-07-10 Молеак Пте Лтд Комбинированная терапия для лечения пациентов с неврологическими нарушениями и церебральным инфарктом
JP2009536660A (ja) * 2006-05-02 2009-10-15 アナコール ファーマシューティカルズ，インコーポレイテッド 加水分解耐性ホウ素含有治療剤及びその使用方法
EP1900378A1 (de) * 2006-08-31 2008-03-19 Novartis AG Pharmazeutische Zusammensetzungen zur Behandlung von Pilzinfektionen
JO3396B1 (ar) * 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc جزيئات صغيرة تحتوي على البورون
JP5504454B2 (ja) * 2007-12-06 2014-05-28 国立大学法人京都大学 新規なホウ素化合物、それらの製造方法およびそれらを用いた機能性電子素子
JP5745279B2 (ja) * 2008-01-09 2015-07-08 アナコール ファーマシューティカルズ，インコーポレイテッド 抗炎症剤としてのホウ素含有小分子
CN102014927A (zh) 2008-03-06 2011-04-13 安纳考尔医药公司 作为抗炎药的含硼的小分子
US20100256092A1 (en) * 2008-05-12 2010-10-07 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010028005A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010027975A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010045503A1 (en) * 2008-10-15 2010-04-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
WO2010044405A1 (ja) 2008-10-15 2010-04-22 キッセイ薬品工業株式会社 縮合環誘導体及びその医薬用途
US8461364B2 (en) * 2008-12-17 2013-06-11 Glaxosmithkline Llc Polymorphs of (S)-3-aminomethyl-7-(3-hydroxy-propoxy)-3H-benzo[C][1,2]oxaborol-1-OL
RU2012107163A (ru) 2009-07-28 2013-09-10 Анакор Фармасьютикалз, Инк. Тризамещенные борсодержащие молекулы
WO2011019618A1 (en) 2009-08-14 2011-02-17 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US20110207701A1 (en) * 2009-08-19 2011-08-25 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011060196A1 (en) 2009-11-11 2011-05-19 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
AP2012006482A0 (en) 2010-03-19 2012-10-31 Anacor Pharmacueticals Inc Boron-containing small molecules as anti-protozoalagent
ES2898695T3 (es) 2010-09-07 2022-03-08 Anacor Pharmaceuticals Inc Derivados de benzoxaborol para el tratamiento de infecciones bacterianas
WO2013050591A2 (en) 2011-10-07 2013-04-11 Syngenta Participations Ag Method for protecting useful plants or plant propagation material
UY34367A (es) * 2011-10-07 2014-08-29 Syngenta Participations Ag ?método para proteger material de propagación vegetal o plantas útiles?.
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
US9138001B2 (en) 2013-01-30 2015-09-22 Agrofresh Inc. Use of benzoxaboroles as volatile antimicrobial agents on meats, plants, or plant parts
US20220125049A1 (en) * 2013-01-30 2022-04-28 Agrofresh Inc. Method and system for centralized management, monitoring, and controlled delivery of biological compounds to fruit storage rooms
WO2014147009A1 (en) * 2013-03-18 2014-09-25 Syngenta Participations Ag Novel microbiocides
WO2014173880A1 (en) 2013-04-22 2014-10-30 Syngenta Participations Ag Novel microbiocides
AU2014202928B1 (en) * 2013-06-05 2014-09-11 Agrofresh Inc. Compounds and compositions
US20170000133A1 (en) * 2013-12-23 2017-01-05 Syngenta Participations Ag Benzoxaborole fungicides
US20170000132A1 (en) * 2013-12-23 2017-01-05 Syngenta Participations Ag Benzoxaborole fungicides
EP3261437B1 (de) * 2015-02-12 2019-09-11 AgroFresh Inc. Fungizide verbindungen und zusammensetzungen
MA41494B1 (fr) * 2015-02-12 2020-10-28 Glaxosmithkline Ip No 2 Ltd Composés benzoxaborole substitués en position 4 et utilisations associées
CN107872956B (zh) * 2015-04-09 2020-07-10 宾夕法尼亚州研究基金会 含有苯并氧杂硼戊环的协同性抗真菌组合物
US10160867B2 (en) * 2015-08-06 2018-12-25 The Penn State Research Foundation Benzoxaborole-containing coating resistant to cellulose-supportable fungus
WO2017031041A1 (en) * 2015-08-17 2017-02-23 Channel Therapeutics, Inc. Functionalized aminobenzoboroxoles
WO2017151489A1 (en) * 2016-03-02 2017-09-08 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
AU2017229096A1 (en) 2016-03-07 2018-09-06 Agrofresh Inc. Vaporized administration of pesticides
TW201735792A (zh) 2016-03-07 2017-10-16 農業保鮮股份有限公司 使用苯并氧雜硼雜環戊烯化合物和防腐氣體作為作物的抗微生物劑之協同方法
US11447506B2 (en) 2016-05-09 2022-09-20 Anacor Pharmaceuticals, Inc. Crystal forms of crisaborole in free form and preparation method and use thereof
CR20180502A (es) 2016-05-12 2018-12-21 Anacor Pharmaceuticals Inc Ésteres de oxaborol y sus usos
US20200262848A1 (en) 2017-11-02 2020-08-20 Halcyon Labs Private Limited Novel process for the preparation tavaborole and its intermediates
JP2021505660A (ja) 2017-11-30 2021-02-18 ボラゲン，インコーポレーテッド ベンゾキサボロール化合物およびその配合物
WO2019173814A1 (en) * 2018-03-09 2019-09-12 University Of The Sciences Protective groups and methods for protecting benzoxaboroles or oxaboroles
WO2020041200A1 (en) 2018-08-18 2020-02-27 Boragen Inc. Solid forms of substituted benzoxaborole and compositions thereof
CN113166177A (zh) 2018-10-05 2021-07-23 辉瑞公司 含硼的pde4抑制剂
US20210024548A1 (en) * 2019-07-25 2021-01-28 Massachusetts Institute Of Technology Boron-containing pharmacophore
AR120504A1 (es) 2019-11-22 2022-02-16 Agrofresh Inc Composición y método para tratar a plantas y partes de plantas con activos volátiles para el control de organismos de descomposición
JP2023512785A (ja) 2020-02-05 2023-03-29 アグロフレッシュ インコーポレイテッド 抗微生物化合物及び組成物
CN114644645B (zh) * 2022-03-08 2023-05-26 南京农业大学 3-吲哚取代苯硼唑类化合物及其制备方法和应用

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Also Published As

Publication number Publication date
CA2190155A1 (en) 1995-12-14
US5880188A (en) 1999-03-09
CN1155286A (zh) 1997-07-23
EP0765331B1 (de) 2000-08-09
WO1995033754A1 (en) 1995-12-14
AU2534895A (en) 1996-01-04
KR970703349A (ko) 1997-07-03
JPH10500983A (ja) 1998-01-27
BR9507966A (pt) 1997-09-02
NO965235L (no) 1997-01-21
GB9411587D0 (en) 1994-08-03
AU681291B2 (en) 1997-08-21
TW368397B (en) 1999-09-01
NO965235D0 (no) 1996-12-06
EP0765331A1 (de) 1997-04-02
CN1068005C (zh) 2001-07-04
ATE195316T1 (de) 2000-08-15
DE69518323D1 (de) 2000-09-14

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee