DE69518323D1 - Oxaborole und deren salze, und deren verwendung als biozide - Google Patents

Oxaborole und deren salze, und deren verwendung als biozide

Info

Publication number
DE69518323D1
DE69518323D1 DE69518323T DE69518323T DE69518323D1 DE 69518323 D1 DE69518323 D1 DE 69518323D1 DE 69518323 T DE69518323 T DE 69518323T DE 69518323 T DE69518323 T DE 69518323T DE 69518323 D1 DE69518323 D1 DE 69518323D1
Authority
DE
Germany
Prior art keywords
pct
oxaborole
biocides
salts
date dec
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69518323T
Other languages
English (en)
Other versions
DE69518323T2 (de
Inventor
William Austin
Juan Kneale
Jelf Crowley
Martin CLOUGH
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Avecia Ltd
Original Assignee
Avecia Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Avecia Ltd filed Critical Avecia Ltd
Application granted granted Critical
Publication of DE69518323D1 publication Critical patent/DE69518323D1/de
Publication of DE69518323T2 publication Critical patent/DE69518323T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • A01N55/08—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur containing boron
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic System
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C08—ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08K—Use of inorganic or non-macromolecular organic substances as compounding ingredients
    • C08K5/00—Use of organic ingredients
    • C08K5/0008—Organic ingredients according to more than one of the "one dot" groups of C08K5/01 - C08K5/59
    • C08K5/0058—Biocides
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09D—COATING COMPOSITIONS, e.g. PAINTS, VARNISHES OR LACQUERS; FILLING PASTES; CHEMICAL PAINT OR INK REMOVERS; INKS; CORRECTING FLUIDS; WOODSTAINS; PASTES OR SOLIDS FOR COLOURING OR PRINTING; USE OF MATERIALS THEREFOR
    • C09D5/00—Coating compositions, e.g. paints, varnishes or lacquers, characterised by their physical nature or the effects produced; Filling pastes
    • C09D5/14—Paints containing biocides, e.g. fungicides, insecticides or pesticides
DE69518323T 1994-06-09 1995-05-26 Oxaborole und deren salze, und deren verwendung als biozide Expired - Fee Related DE69518323T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9411587A GB9411587D0 (en) 1994-06-09 1994-06-09 Compound, composition and use
PCT/GB1995/001206 WO1995033754A1 (en) 1994-06-09 1995-05-26 Oxaboroles and salts thereof, and their use as biocides

Publications (2)

Publication Number Publication Date
DE69518323D1 true DE69518323D1 (de) 2000-09-14
DE69518323T2 DE69518323T2 (de) 2001-02-01

Family

ID=10756481

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69518323T Expired - Fee Related DE69518323T2 (de) 1994-06-09 1995-05-26 Oxaborole und deren salze, und deren verwendung als biozide

Country Status (14)

Country Link
US (1) US5880188A (de)
EP (1) EP0765331B1 (de)
JP (1) JPH10500983A (de)
KR (1) KR970703349A (de)
CN (1) CN1068005C (de)
AT (1) ATE195316T1 (de)
AU (1) AU681291B2 (de)
BR (1) BR9507966A (de)
CA (1) CA2190155A1 (de)
DE (1) DE69518323T2 (de)
GB (1) GB9411587D0 (de)
NO (1) NO965235L (de)
TW (1) TW368397B (de)
WO (1) WO1995033754A1 (de)

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KR101337068B1 (ko) * 2005-02-16 2013-12-06 아나코르 파마슈티칼스 인코포레이티드 보론함유 소분자
CN102532180B (zh) * 2005-12-30 2016-06-29 安纳考尔医药公司 含硼的小分子
JP2009526751A (ja) 2005-12-30 2009-07-23 アナコール ファーマシューティカルズ，インコーポレイテッド ホウ素含有小分子
EP1988779B1 (de) 2006-02-16 2015-06-24 Anacor Pharmaceuticals, Inc. Kleine boronhaltige moleküle als entzündungshemmende wirkstoffe
US20070197388A1 (en) * 2006-02-22 2007-08-23 Buckman Laboratories International, Inc. Haloperoxidase treatment to control algae
AU2007225456B2 (en) * 2006-03-16 2013-03-28 Moleac Pte Ltd Combination therapy for treatment of patients with neurological disorders and cerebral infarction
WO2007131072A2 (en) * 2006-05-02 2007-11-15 Anacor Pharmaceuticals, Inc. Hydrolytically-resistant boron-containing therapeutics and methods of use
EP1900378A1 (de) * 2006-08-31 2008-03-19 Novartis AG Pharmazeutische Zusammensetzungen zur Behandlung von Pilzinfektionen
JO3396B1 (ar) * 2007-06-20 2019-10-20 Anacor Pharmaceuticals Inc جزيئات صغيرة تحتوي على البورون
JP5504454B2 (ja) * 2007-12-06 2014-05-28 国立大学法人京都大学 新規なホウ素化合物、それらの製造方法およびそれらを用いた機能性電子素子
JP5745279B2 (ja) * 2008-01-09 2015-07-08 アナコール ファーマシューティカルズ，インコーポレイテッド 抗炎症剤としてのホウ素含有小分子
US8039450B2 (en) 2008-03-06 2011-10-18 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
EP2285384A4 (de) * 2008-05-12 2012-04-25 Anacor Pharmaceuticals Inc Borhaltige kleine moleküle
WO2010028005A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010027975A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2010045503A1 (en) 2008-10-15 2010-04-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agents
MX2011004088A (es) 2008-10-15 2011-09-06 Kissei Pharmaceutical Derivado de anillo fusionado y su aplicacion medica.
AU2009335744A1 (en) 2008-12-17 2010-07-15 Anacor Pharmaceuticals, Inc. Polymorphs of (S)-3-aminomethyl-7-(3-hydroxy-propoxy) -3H-benzo[c][1,2] oxaborol-1-ol
US8343944B2 (en) 2009-07-28 2013-01-01 Anacor Pharmaceuticals, Inc. Trisubstituted boron-containing molecules
WO2011019618A1 (en) 2009-08-14 2011-02-17 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011022337A1 (en) * 2009-08-19 2011-02-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US9346834B2 (en) 2009-10-20 2016-05-24 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
US8461134B2 (en) 2009-11-11 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011094450A1 (en) 2010-01-27 2011-08-04 Anacor Pharmaceuticals, Inc Boron-containing small molecules
US8623911B2 (en) 2010-03-19 2014-01-07 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
DK3251678T3 (da) 2010-09-07 2021-11-22 Anacor Pharmaceuticals Inc Benzoxaborolderivater til behandling af bakterieinfektioner
EP2763538A2 (de) * 2011-10-07 2014-08-13 Syngenta Participations AG Verfahren zum schützen von nutzpflanzen oder pflanzenpropagierungsmaterial
UY34367A (es) * 2011-10-07 2014-08-29 Syngenta Participations Ag ?método para proteger material de propagación vegetal o plantas útiles?.
US9585396B2 (en) 2013-01-30 2017-03-07 Agrofresh Inc. Volatile applications against pathogens
US8669207B1 (en) 2013-01-30 2014-03-11 Dow Agrosciences, Llc. Compounds and compositions
US11039617B2 (en) 2013-01-30 2021-06-22 Agrofresh Inc. Large scale methods of uniformly coating packaging surfaces with a volatile antimicrobial to preserve food freshness
US20220125049A1 (en) * 2013-01-30 2022-04-28 Agrofresh Inc. Method and system for centralized management, monitoring, and controlled delivery of biological compounds to fruit storage rooms
CA2899317A1 (en) * 2013-01-30 2014-08-07 Dow Agrosciences Llc Use of benzoxaboroles as volatile antimicrobial agents on meats, plants, or plant parts
US10070649B2 (en) 2013-01-30 2018-09-11 Agrofresh Inc. Volatile applications against pathogens
WO2014147009A1 (en) * 2013-03-18 2014-09-25 Syngenta Participations Ag Novel microbiocides
WO2014173880A1 (en) 2013-04-22 2014-10-30 Syngenta Participations Ag Novel microbiocides
AU2014202928B1 (en) * 2013-06-05 2014-09-11 Agrofresh Inc. Compounds and compositions
EP3086644A1 (de) * 2013-12-23 2016-11-02 Syngenta Participations AG Benzoxaborolfungizide
WO2015097276A1 (en) * 2013-12-23 2015-07-02 Syngenta Participations Ag Benzoxaborole fungicides
MA41494B1 (fr) * 2015-02-12 2020-10-28 Glaxosmithkline Ip No 2 Ltd Composés benzoxaborole substitués en position 4 et utilisations associées
MX2017010302A (es) * 2015-02-12 2017-12-07 Agrofresh Inc Compuestos y composiciones fungicidas.
EP3280262B1 (de) * 2015-04-09 2022-07-06 The Penn State Research Foundation Fungizide zusammensetzung mit synergistischem benzoxaborol
WO2017024022A1 (en) * 2015-08-06 2017-02-09 The Penn State Research Foundation Benzoxaborole-containing coating resistant to cellulose-supportable fungus
US10633399B2 (en) 2015-08-17 2020-04-28 Channel Therapeutics, Inc. Functionalized aminobenzoboroxoles
CN109195608B (zh) * 2016-03-02 2021-05-11 比尔及梅琳达盖茨基金会 含硼小分子
NZ745681A (en) 2016-03-07 2022-05-27 Agrofresh Inc Synergistic methods of using benzoxaborole compounds and preservative gases as an antimicrobial for crops
TW201733442A (zh) 2016-03-07 2017-10-01 農業保鮮股份有限公司 殺有害生物劑之汽化給予
US11447506B2 (en) 2016-05-09 2022-09-20 Anacor Pharmaceuticals, Inc. Crystal forms of crisaborole in free form and preparation method and use thereof
KR102243775B1 (ko) 2016-05-12 2021-04-22 아나코르 파마슈티칼스 인코포레이티드 옥사보롤 에스터 및 이의 용도
EP4119566A1 (de) 2017-11-02 2023-01-18 Halcyon Labs Private Limited Neues verfahren zur herstellung von tavaborol und dessen zwischenprodukten
BR112020010927A2 (pt) 2017-11-30 2020-12-01 Boragen, Inc. compostos de benzoxaborol e formulações dos mesmos
WO2019173814A1 (en) 2018-03-09 2019-09-12 University Of The Sciences Protective groups and methods for protecting benzoxaboroles or oxaboroles
EP3836938A4 (de) * 2018-08-18 2022-05-11 Boragen, Inc. Feste formen von substituiertem benzoxazol und zusammensetzungen davon
PE20211546A1 (es) 2018-10-05 2021-08-16 Pfizer Inhibidores de pde4 que contienen boro
US20210024548A1 (en) * 2019-07-25 2021-01-28 Massachusetts Institute Of Technology Boron-containing pharmacophore
AR120504A1 (es) 2019-11-22 2022-02-16 Agrofresh Inc Composición y método para tratar a plantas y partes de plantas con activos volátiles para el control de organismos de descomposición
PE20221733A1 (es) * 2020-02-05 2022-11-07 Agrofresh Inc Composiciones y composiciones antimicrobianas
CN114644645B (zh) * 2022-03-08 2023-05-26 南京农业大学 3-吲哚取代苯硼唑类化合物及其制备方法和应用

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Also Published As

Publication number Publication date
JPH10500983A (ja) 1998-01-27
DE69518323T2 (de) 2001-02-01
BR9507966A (pt) 1997-09-02
CN1155286A (zh) 1997-07-23
EP0765331A1 (de) 1997-04-02
KR970703349A (ko) 1997-07-03
EP0765331B1 (de) 2000-08-09
NO965235D0 (no) 1996-12-06
CA2190155A1 (en) 1995-12-14
ATE195316T1 (de) 2000-08-15
AU2534895A (en) 1996-01-04
AU681291B2 (en) 1997-08-21
CN1068005C (zh) 2001-07-04
WO1995033754A1 (en) 1995-12-14
US5880188A (en) 1999-03-09
NO965235L (no) 1997-01-21
GB9411587D0 (en) 1994-08-03
TW368397B (en) 1999-09-01

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee