DE60122193D1 - Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten - Google Patents

Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten

Info

Publication number
DE60122193D1
DE60122193D1 DE60122193T DE60122193T DE60122193D1 DE 60122193 D1 DE60122193 D1 DE 60122193D1 DE 60122193 T DE60122193 T DE 60122193T DE 60122193 T DE60122193 T DE 60122193T DE 60122193 D1 DE60122193 D1 DE 60122193D1
Authority
DE
Germany
Prior art keywords
glucopyranosyloxybenzylbenzen
derivatives
compounds
compositions containing
medical compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60122193T
Other languages
English (en)
Other versions
DE60122193T2 (de
Inventor
Nobuhiko Fushimi
Toshihiro Nishimura
Kazuya Tatani
Masayuki Isaji
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kissei Pharmaceutical Co Ltd
Original Assignee
Kissei Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kissei Pharmaceutical Co Ltd filed Critical Kissei Pharmaceutical Co Ltd
Publication of DE60122193D1 publication Critical patent/DE60122193D1/de
Application granted granted Critical
Publication of DE60122193T2 publication Critical patent/DE60122193T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/203Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
DE60122193T 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten Expired - Lifetime DE60122193T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2000301523 2000-09-29
JP2000301523 2000-09-29
PCT/JP2001/008239 WO2002028872A1 (fr) 2000-09-29 2001-09-21 Derives de glucopyranosiloxybenzylbenzene et compositions therapeutiques contenant ces composes

Publications (2)

Publication Number Publication Date
DE60122193D1 true DE60122193D1 (de) 2006-09-21
DE60122193T2 DE60122193T2 (de) 2007-07-05

Family

ID=18783054

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60122193T Expired - Lifetime DE60122193T2 (de) 2000-09-29 2001-09-21 Glucopyranosyloxybenzylbenzol derivate und medizinische zusammensetzungen, die diese verbindungen enthalten

Country Status (33)

Country Link
US (2) US6872706B2 (de)
EP (1) EP1329456B1 (de)
JP (1) JP3798375B2 (de)
KR (1) KR100647204B1 (de)
CN (1) CN1293087C (de)
AR (1) AR030816A1 (de)
AT (1) ATE335753T1 (de)
AU (2) AU9025701A (de)
BG (1) BG66015B1 (de)
BR (1) BR0114310A (de)
CA (1) CA2423568C (de)
CY (1) CY1106076T1 (de)
CZ (1) CZ303544B6 (de)
DE (1) DE60122193T2 (de)
DK (1) DK1329456T3 (de)
EA (1) EA005994B1 (de)
ES (1) ES2269456T3 (de)
HK (1) HK1061037A1 (de)
HU (1) HUP0301178A3 (de)
IL (2) IL155071A0 (de)
MX (1) MXPA03002779A (de)
MY (1) MY129023A (de)
NO (1) NO327182B1 (de)
NZ (1) NZ524917A (de)
PE (1) PE20020476A1 (de)
PL (1) PL205607B1 (de)
PT (1) PT1329456E (de)
SI (1) SI1329456T1 (de)
SK (1) SK287811B6 (de)
TW (1) TWI284641B (de)
UA (1) UA73606C2 (de)
WO (1) WO2002028872A1 (de)
ZA (1) ZA200302283B (de)

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WO2004050122A1 (ja) * 2002-12-04 2004-06-17 Kissei Pharmaceutical Co., Ltd. 高血糖症に起因する疾患の予防又は治療剤
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DE10258008B4 (de) * 2002-12-12 2006-02-02 Sanofi-Aventis Deutschland Gmbh Heterocyclische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel
DE10258007B4 (de) * 2002-12-12 2006-02-09 Sanofi-Aventis Deutschland Gmbh Aromatische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel
UA86042C2 (en) * 2003-08-01 2009-03-25 Янссен Фармацевтика Н.В. Substituted indazole-o-glucosides
EP2360164A3 (de) * 2004-03-16 2012-01-04 Boehringer Ingelheim International GmbH Glucopyranosyl-substituierte Benzol-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
US20070185197A1 (en) * 2004-03-31 2007-08-09 Hideki Fujikura Phenol derivative, medicinal composition containing the same, and medicinal use thereof
ES2581331T3 (es) * 2004-07-21 2016-09-05 Kissei Pharmaceutical Co., Ltd. Inhibidor de la progresión de una enfermedad atribuida a una acumulación anormal de grasa hepática
TW200606129A (en) 2004-07-26 2006-02-16 Chugai Pharmaceutical Co Ltd Novel cyclohexane derivative, its prodrug, its salt and diabetic therapeutic agent containing the same
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UA91546C2 (uk) 2005-05-03 2010-08-10 Бьорінгер Інгельхайм Інтернаціональ Гмбх КРИСТАЛІЧНА ФОРМА 1-ХЛОР-4-(β-D-ГЛЮКОПІРАНОЗ-1-ИЛ)-2-[4-((S)-ТЕТРАГІДРОФУРАН-3-ІЛОКСИ)-БЕНЗИЛ]-БЕНЗОЛУ, СПОСІБ ЇЇ ОДЕРЖАННЯ ТА ЇЇ ЗАСТОСУВАННЯ ПРИ ПРИГОТУВАННІ ЛІКАРСЬКИХ ЗАСОБІВ
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UA97817C2 (ru) 2006-12-06 2012-03-26 Глаксосмиткляйн Ллк Гетероциклические производные 4-(метилсульфонил)фенила и их применение
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Also Published As

Publication number Publication date
AR030816A1 (es) 2003-09-03
MY129023A (en) 2007-03-30
NZ524917A (en) 2005-01-28
CA2423568C (en) 2011-03-15
EP1329456A1 (de) 2003-07-23
HUP0301178A3 (en) 2009-08-28
DK1329456T3 (da) 2006-12-04
CN1466590A (zh) 2004-01-07
BG107674A (bg) 2004-01-30
SI1329456T1 (sl) 2006-12-31
BG66015B1 (bg) 2010-10-29
ATE335753T1 (de) 2006-09-15
PL362177A1 (en) 2004-10-18
EA005994B1 (ru) 2005-08-25
BR0114310A (pt) 2003-10-14
JP3798375B2 (ja) 2006-07-19
WO2002028872A1 (fr) 2002-04-11
HUP0301178A2 (hu) 2003-11-28
US20040018998A1 (en) 2004-01-29
AU2001290257B2 (en) 2007-08-30
EA200300316A1 (ru) 2003-08-28
US6872706B2 (en) 2005-03-29
EP1329456B1 (de) 2006-08-09
IL155071A (en) 2010-04-15
NO20031407L (no) 2003-04-30
US20050065098A1 (en) 2005-03-24
TWI284641B (en) 2007-08-01
ZA200302283B (en) 2005-05-27
PT1329456E (pt) 2006-12-29
CZ303544B6 (cs) 2012-11-28
KR20030036867A (ko) 2003-05-09
CA2423568A1 (en) 2002-04-11
AU9025701A (en) 2002-04-15
CN1293087C (zh) 2007-01-03
IL155071A0 (en) 2003-10-31
HK1061037A1 (en) 2004-09-03
CY1106076T1 (el) 2011-06-08
UA73606C2 (en) 2005-08-15
PE20020476A1 (es) 2002-07-04
JPWO2002028872A1 (ja) 2004-02-12
PL205607B1 (pl) 2010-05-31
EP1329456A4 (de) 2005-03-30
ES2269456T3 (es) 2007-04-01
DE60122193T2 (de) 2007-07-05
MXPA03002779A (es) 2004-05-04
KR100647204B1 (ko) 2006-11-17
NO20031407D0 (no) 2003-03-27
SK3342003A3 (en) 2003-08-05
NO327182B1 (no) 2009-05-04
SK287811B6 (sk) 2011-10-04

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